Ola kino, Hoomakaukau
"Felodip": aʻo no ka hoʻohana, nāʻana. lāʻau analogues
I kahea aku nei oia no ka lāʻau "Felodip"? Na Ke Kumu no ka hoʻohana ana i ka lāʻau, e e ho'ākāka 'ia ma ka au mamuli o ka hooku iho la ia pauku. No hoi kekahi poe mai o ia, oe, e aʻo e pili ana i mea keia k ua ia, ahaʻaoʻao 'ole ka mea, ua loaa, ina paha i keia k contraindications, pehea ka nui o ka mea, na koina, i mea analogues, a pela aku.
I ka haku mele 'ana o ka lāʻau, i ka palapala o ka manufacturing, a me ka'ōpala
Ma ka palapala hiki ke loaʻa ma ka hale kūʻai lāʻau lapaʻau lāʻau "Felodip"? ma o ka hana o keia ka lapaʻauʻia alakai hākālia nō i ka mea i loaʻa i loko o ka palapala o ka papa me ka hooloihi ae i hana wale. A,ʻokoʻa nā māhele o ka lāʻau i kaʻokoʻa wahī:
- yellow huaale i loko o ka palapala o ka papapa, me kekahi ala denoted ma ka helu 2,5. Kaʻeleu hehee ai ka lāʻau felodipine hana i loko o ka nui o 2,5 mg. Excipients o ka lāʻau i lactose monohydrate, hypromellose, microcrystalline kelulose, ula hao'okesaside, povidone, titanium'okikene lua, propyl gallate, lenalena hao'okesaside, makanekiuma stearate, propylene glycol, anhydrous colloidal ka silica i, talc. Ma ke kuai ana o ka hana lāʻau komo ka blister 10 papa i i waihoia ma ka pepa pahu.
- O na papa io o ka malamalama a pink ano i loko o ke kinona o ka papapa, me kekahi ala denoted ma ka helu 5. Kaʻeleu ke keʻena o ka la hoomalolo protrudes felodipine i loko o ka nui o ka 5 mg. Excipients o ka lāʻau nei iluna lactose monohydrate, hypromellose, microcrystalline kelulose, ula hao'okesaside, povidone, titanium'okikene lua, propyl gallate, lenalena hao'okesaside, makanekiuma stearate, propylene glycol, anhydrous colloidal ka silica i, talc. Ma ke kuai ana o ka hana lāʻau komo ka blister 10 na papa, e hoonoho iho i ka pepa pahu.
- Papa ulaula iki eleele papapa hoʻokino me kekahi ala i koho numeral 10. kaʻeleu hehee ai o ia i ka lāʻau felodipineʻoihana'ē aʻe i loko o ka nui o ka 10 mg. Auxiliaries i lactose monohydrate, hypromellose, microcrystalline kelulose, ula hao'okesaside, povidone, titanium'okikene lua, propyl gallate, lenalena hao'okesaside, makanekiuma stearate, propylene glycol, anhydrous colloidal ka silica i, talc. Ma ke kuai ana o ka hana lāʻau komo ka blister 10 papa. Blisters kau i ka pepa pahu.
Ke pharmacological waiwai o ka lāʻau
He aha mea he 'inikua mea "Felodip"? Na Ke Kumu no ka hoʻohana ana i ka lāʻau 'mai nei ia ia mea i ke kalipuna Kanal blocker lohi. Nānā akula au i ka lāʻau 'no a hiki i ka pae o ka dihydropyridine.
Kēia ka lapaʻauʻia mea hiki ke kulia antianginal a me ka antihypertensive 'ole. Eia hou, e ho'ēmi i kā ka'aloʻahiʻa (koko) ma ka hōʻemiʻanaʻike ākea vascular e kū'ē'ē mai.
He aha nā waiwai i ai ' "Felodip"? Na Ke Kumu no ka hoʻohana ana i ka la hoomalolo kikowaena ike ana ia i paʻa i ka mahele lāʻau-e kaukaʻi Anati-ischemic hopena. Ka lapaʻauʻia ho'ēmi i kā infarction nui, a hoi i malama i ke kino, mai reperfusion complications.
Kēia mea paahana i kokoke ole io inotropic hopena. Ua loaʻa he ka palena haʻahaʻa hopena ma luna o ka hoʻokō 'ia' nenoaiu.
Nā pharmacokinetics o ka lāʻau
Pehea lā ka lōʻihi o ka lāʻau o ke kemu, "Felodip"? Na Ke Kumu no ka hoʻohana 'ana, ua manaʻo' o ia hoʻi i ka mea ma hope o ka mahele lāʻau o medicament i loko o kaʻeleu waiwai ua kokoke loa ke kemu, mai ka digestive'āpana, a hana koke. Mahalo i kona laʻau heluna ano, lohi kala o kaʻeleu hehee ai e hōʻoiaʻiʻo konaʻaʻahu lehulehu i loko o ke koko (i loko o ka lā), a me hiki aku ai i ka hua i loko o ka omo pae.
Mākou hiki ole ke olelo i ka bioavailability o ka lāʻau, aole ia e hilinaʻi ma ka pākōlea mahele lāʻau a me ka mea o ka hola 15%.
Paa i ka wai koko nā polokina, a oi kaʻoi loa ia mea o ka hola 99%. Ua hookuu a ke medicament me ka umauma waiu, a komo iloko o ke koko-lolo ke'ākeʻakeʻa mai, a me ka placental ke'ākeʻakeʻa mai. Me ka hooloihi ae i hoʻohana ana i ka hana waiwai ole hoʻomāhuahua ia lŘlŘ.
Where ka lāʻau ua metabolized "Felodip"? Kaʻeleu 'Oponopono o keia Agena ua metabolized ma ke akepaʻa. Ma keia palapala AEeOEXAaI metabolites.
Ka hapa-ola o ka lāʻau ma kahi o ka 25 hola. E hōʻike 'makaukau like metabolites (ka hola 70%) i loko o ka mimi a me feces (30%).
nāʻikepili medicament
Ma kekahi mau hihia, i ka hoʻomanawanui ua hoakakaia ka lapaʻauʻia "Felodip" (5 mg) Na Ke Kumu o keia ka lapaʻauʻia loaʻa nā kēia papa inoa o nāʻikepili no ka i:
- hypertension;
- angina;
- arrhythmia;
- coronary naau maʻi;
- circulatory kāna hana;
- Raynaud ka maʻi pale.
Contraindications ai '
Ma i na hihia ua pololei papaia e lawe ka lapaʻauʻia "Felodip"? Reviews o nā kauka, e like me ka mea hele pū ana me ka olelo hoakaka e ole e hoʻohana 'ia ka lāʻau ma lalo o ke ana ma lalo nei:
- huʻi myocardial infarction, e like me loko o hoʻokahi mahina ma hope o myocardial;
- lolelua ka angina;
- cardiogenic kŰia;
- naau ole, o ka oi aku decompensated;
- aortic stenosis (clinically nui);
- hāpai keiki;
- hypotension (loa);
- i loko o nā keiki a me nā adolescents (ma lalo makahiki 18);
- i lactation;
- mahuahua pā lonoaʻili o ka hoʻomanawanui a hiki i ka lāʻau a mea 'ē aʻe dihydropyridine nā mea loaʻa.
Kekahi e mai poina i keia koʻi me ka lōʻihi mālama nui i hoakaka ia i nā mea maʻi me ka hepatic a me kaʻaʻa puʻuwai insufficiency.
Lapaʻau mea hoʻoluku "Felodip": kauoha no ka hoʻohana
Analogues o keia mea paahana, e ia ke hōʻike i ka iki ae la. Ano, au makemake e hai aku ia oe e pili ana pehea e e lawe pololei 'ia o ka lapaʻauʻia.
I ka hypertension mahele lāʻau no nā mākua a me ka poʻeʻelemākule e ua waiho pākahi. Nō kāu, i ka loiloi mua dala o ka lāʻau, he 5 mg koke i ka lā. Ma ke koho ana i kūpono e hoomanawanui i ka laʻau heluna ua waiho e hoʻohana i ka papa o 2,5 mg. A hiki aku i ka manaʻo pono, e hoomahuahua i ka mahele lāʻau o ka lapaʻauʻia hiki ia. Ka awelika ka leo o ka medicament no ka mālama 'ana i iapaau ana o 5-10 mg no ka lā.
No ka poʻeʻelemākule nā mea maʻi a me nā mea maʻi me ka hihia ake hana ma ke kakahiaka lāʻau Inc ua lawelawe i loko o ka nui o ka 2,5 mg no ka lā.
Ma ka pilina paʻa angina lapaau "Felodip" i kuhikuhi pākahi. Pela o ka puka mua mahele lāʻau (no nā mākua) mea 5 mg koke i ka lā. Inā koi 'ia, hiki e mahuahua ai ka mahele lāʻau a hiki i 10 mg no ka lā. ʻO kā mākou kela la i keia dala o ka lāʻau, he 20 mg.
Papa "Felodip" ua aeia mai e lawe i ka hui pu ana, me ka ACE nā mea kūpale, Hoʻokolohua-blockers a me diuretics. Naʻe, ka mea e e hoʻomaopopo i oiai ka hypotensive hopena ua hoʻokāʻoi '. No ia mea, e pono e loa makaala no ka mea, o ka mahuahua kamepiula o ke hypotension.
Ma nā mea maʻi me ka loa hihia hoʻi ake hana e hoemi i ka mahele lāʻau o ka lapaʻauʻia e.
I hoʻouna 'ia ma ka lāʻau e wale e ia i loko o ke kakahiaka mua aina kakahiaka. Ma keia hihia, no ka papa ma kekahi hihia he mea hiki ole ke crack, e hoea a māhele.
overdose ano
Pololei ole 'ana o nā huaale "Felodip" na kēia symptoms o overdose kānāwai i loko o nā mea maʻi: bradycardia a me ka hypotension (loa).
I Ina o ka hanana o ia mau symptoms symptomatic Inc. Inā hypotension (loa) nā mea maʻi e haawi aku i ka papamoeʻoihana, a hookiekie ae wāwae. Me ka mahalo i ka bradycardia, ma a ina o ka hoʻomanawanui atropine lawelawe intramuscularly ma ka laʻau heluna o 0.5-1 mg. Inā pono, e hoomahuahua i ka buke o ka wai koko infusion ua lawe mai me ka paʻakai koloriside, monakō koko pāʻoihana a me dextran.
I ka wa a ka luna-i ho'ākāka 'ia inefficiency ana i koi' ia ka lapaʻauʻia i ka hoomanawanui me ka predominant ia ma Alpha-adrenergic receptors.
ʻaoʻao 'ole, mai ka lalau ana i ka lāʻau'
E hiki anei i ka hopena maikaʻi 'ole ma o ka kanaka kino e lawe i ka lapaau "Felodip"? Analogues o keia mea paahana, a hoomakaukau iho pinepine ke kumu no headache, lehalehu t flushing, pōniuniu, palpitations a me ka luhi. Naʻe, ka mea e e kaulana i ka reactions i reversible. Ka mea, i hookuu hou i ka hoʻomaka o ka Inc, e like me ma ka hoʻoulu i ka laʻau heluna o ka lāʻau.
Ma ke alanui, ke kaumaha ma muli o ka nui i loaa ka lapaʻauʻia ka hoʻomanawanui iʻikea a me kaʻike ākea edema. E like me ka poe akamai, ka mea, i ka hopena o precapillary vasodilation.
Ma nā mea maʻi me ka periodontal a nui aʻe ana mai i loko o nā mea maʻi e loaa ana i ka lāʻau 'i ia he uuku nani o ka nui aʻe ana. Kēia kaʻina hana hiki e Hāʻule maila lākou, ina oe e malama hoʻokolokolo pono ku una kou niho.
Ma kekahi hihia mākou e noʻonoʻo 'ana i ka loaa ana ka lapaʻauʻia i ke kumu o ka kēiaʻaoʻao ole:
- Mea'ōnaehana mānowai koko'ōnaehana: palpitations, tachycardia, a me kaʻike ākea edema.
- Dermatological reactions: photosensitivity, pruritus, urticaria.
- ʻike ākea a Central ko mākou hopohopo'ōnaehana: paresthesia, headache a me ka pōniuniu.
- Musculoskeletal'ōnaehana: arthralgia, myalgia.
- Digestive'āpana: gingival hyperplasia, nausea, hoomahuahua i ake nā'ūhū.
- Other: luhi, hypersensitivity reactions, me angioedema.
Analogs, a me ka waiwai e lilo aku ana i ka lāʻau '
Pehea ka nui o ka lapaʻauʻia ma mua iā mākou? Ia mea i ka hihia ma na mea he nui nā mea maʻi undergoing keia iapaau ana i ka lawelawe. It E e kaulana ia keia mea he lapaau hiki ke kuai i ke kēia kala:
- O na papa io o ka 2,5 mg (30 na apana) - 425 Lūkini rubles;
- papa i loko o ka buke o ka 5 mg (30 na apana) - 556 Lūkini rubles;
- huaale i loko o ka buke o ka 10 mg (30 na apana) - 831 Lūkini rubles.
He aha e puku i ka lāʻau "Felodip"? i loaʻa Analogs o keia k ma kaʻaneʻane nā hale kūʻai lāʻau lapaʻau. Iwaena o lakou, au makemake e kahińuli i ka keia mau laau:. "Plendil," "Felodipine-NW", "Felodipine" a me ka "Felotenz retard"
Maikaʻi i kou manaʻo, mai nā mea maʻi e pili ana i lāʻau lapaʻau huahana
Hoike e pili ana i "Felodip" hoomakaukau moku'āina i ia mea i aloha pono a me ka maikaʻi-tolerated e hoʻomanawanui iki mai, nānā 'ole o ka makahiki a me ka ka wahine. Eia kekahi,ʻeleu lāʻau hiki ke laweia'ku ko e hoʻomanawanui iki mai me ka mimikō,ʻaʻa puʻuwai kāna hana, asthma a me nā obstructive akemāmā maʻi me Raynaud ka maʻi pale, hyperlipidemia, gout, a ma hope o akemāmā transplantation.
Ua nui na poe akamai i kuhikuhi mai i ka mea i ka laau lapaau i ole ia ma ka lipid holoʻokoʻa a me ke koko monakō koko lehulehu.
hopena maikaʻi 'hōʻike manaʻo
Mawaena o ka hopena maikaʻi hōʻike manaʻo e haʻalele nā mea maʻi ma luna o keia k, ua hiki e hoailona oukou ka poe i pili i ka mea kiʻekiʻe lilo o ka lāʻau. ʻOiai pharmacists hoʻopaʻapaʻa ana i kona kumukuai mea oo pahuhopu nei me ka hoʻokōʻana a me ka mea e like ai.
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