Ola kinoHoomakaukau

"Losek CI": olelo ao no ka hoʻohana. "Losek CI": lapaʻau, nāʻana, nāʻikepili, contraindications

Anei oe i ike o ka mea, mai ka mea i kēia lāʻau 'like "Losek CI"? Na Ke Kumu no ka hoʻohana 'ana, e like me nāʻikepili o ka lāʻau, e e ho'ākāka' ia i loko o kēia 'atikala. Eia hou, e hōʻike mākou oe i ka nui o ia na koina, i mai la mea, ina loaa ia ia kekahi analogues a me contraindications, kaʻaoʻao 'ole ana ma hope o ka hoʻoponopono, a me ka oi.

Haku mele 'ana, a me ka'ōpala ke ano o ka lāʻau

He aha mea i ka laau "Losek CI"? Na Ke Kumu no ka hoʻohana hoʻomaopopo 'o ia iā mākou i kēia k mea loaʻa wale nō ma ka papa palapala. Kaʻeleu hehee ai medicament hana omeprazole (10, 40 a me 20 mg). No hoi o na papa io nā a kākoʻo nā mea hoʻohui: glyceryl monostearate, MCC, hydroxypropylmethylcellulose, hydroxypropylcellulose, makanekiuma stearate, kōpaʻa, methacrylicʻakika, talc, paraffin, triethyl citrate, polyethylene glycol, titanium'okikene lua, polysorbate, hao'okesaside, crosslinked polyvinylpyrrolidone a me ka paʻakai stearyl fumarate .

Kūʻai 'medicament i ia i loko o ka hue ili o 14, 7 a me 28 o na papa io (10, 40 a me 20 mg) Ua waiho ia ma ka pepa pahu.

pharmacodynamics

Pehea ke ano o ka lāʻau "Losek CI"? Na Ke Kumu no ka hoʻohana Hawaii iʻeleu lāʻau mea he inhibitor o ka H + -K + -ATPase. Eia hoʻi, ka mea pili i ka Anati-ulcer konohiki. Konaʻeleu Agena mea he nawaliwali kumu. Ua ua i kia ma kaʻakika 'ia o ka parietal keena o ka gastric mucosa, ho'ā' ia paha, a inhibiting ka proton EII ni.

Kanawai o omeprazole ma luna o ka mea i ho'ākāka 'ia kaʻina mea mahele lāʻau-e kaukaʻi. A medicament hiki ke hoʻolako 'nui ka hoʻokō inhibition o basal a hauma¯naʻakika secretion irrespective o ka stimulatory ololi.

Kanawai ma ka secretion o gastric wai

Me kela la i keia moʻolelo medicament "Losek CI", ke kumukuai o ka mea e e imua i iki aku, ua hoakaka pono a me ka kokololio inhibition o nighttime a me ka ao, secretion o hydrochloricʻakika. Ka nui pākōlea hopena ua malama i loko o 4 lā o ka nohoʻana. People me ka ulcer 12 duodenal ulcer 20 mg o ka lāʻau ke kumu i ka napoo ka ho'ēmiʻana i loko o 24-hora gastricʻakika o ole e emi malalo o 80%. It E e kaulana no hoi i keia mahele lāʻau o ka medicament mea hiki ke malama i ka meakino i loko o intragastricʻakika kiʻekiʻe o ka pH> 3. Ua like me ia mau no ka 17 hola.

Ole ma Helicobacter pylori

Pehea ka pono hana ku ei ka olelo mai koʻohune lapaau "Losek CI"? Ka hooponopono hoohui ana i ka lāʻau, wahi a ua omeprazole i ke kiʻekiʻe bactericidal ia ma Helicobacter pylori. Eradication o koʻohune i ka palapala o ia hoʻi, ma ka hui pu ana, me ka Anati-mea koʻohune ai 'ua pu ma ka' ano kokololio hoʻopau o nā symptoms, e like me keʻano kiʻekiʻe o ka hoola ana mai o ka loli ana o mucosa o ka digestive'āpana. Eia hou, ua iapaau ana paipai 'ia ka lōʻihi-makahiki ke kala ana o ka ulcerative maʻi, a me ka nui loa ho'ēmi i kā ka likelihood o recurrent kahe ana ke koko.

Other waiwai o ka lāʻau

He aha nā waiwai i ka hoʻomākaukau me "Losek CI"? House poe akamai i stipulate e hoʻomanawanui iki mai i mau, a no ka lōʻihi manawa, lawe lapaʻauʻia e emi i ka secretion o na glands o ka digestive'āpana, ka mea, ua pinepine malama glandular cysts i loko o ka'ōpū. E like me ka rula, ka mea, ua benign, a nalo ma luna o lākou iho.

Hakumakuma o hydrochloricʻakika secretion i loko o ka'ōpū paipai 'ia ka maʻamau intestinal microflora. Naʻe, i kēia e alakai i ka hōʻemi iki ulu i loko o ka pilikia o ka ulu nā mea palahēhē.

Ma nā mākua a me nā keiki, lōʻihi-makahiki lawe ia ana o na dala, i ka mea ulu ma ka helu o enterochromaffin keena malama.

Ma lapaʻau me omeprazole lehulehu o gastrin i loko o ke koko me ka nui loa māhuahua.

Pharmacokinetics

Komo ka paka i loko o ke koko ka lapaʻauʻia "Losek CI"? Na Ke Kumu no ka hoʻohana hoʻike i omo o ka omeprazole ia lŘlŘ ma ka liʻiliʻi liʻiliʻi (i loko o 4-6 hola). Palaoa ma luna o ka bioavailability o ka waiwai a ua i loli. Ma hope o moʻolelo aaieieno? Ia mea ma kahi o 60%.

Ka lāʻau 'ua loa metabolized ma ke akepaʻa. Ka hapa-ola nei ma kahi o 30-80 minuke. Kahi o 80% o kaʻeleu waiwai ua excreted like metabolites ma nā puʻupaʻa, a me ke koena a me ka feces.

hoike

Papa "Losek CI" ua hoakaka no ka mea kēia deviations:

  • houpo ulcer;
  • reflux esophagitis;
  • ulcer 12 duodenal ulcer;
  • ka'aʻaiawāʻana o ka naʻau liʻiliʻi, kena ae la ia e NSAIDs;
  • eradication o Helicobacter pylori;
  • dyspepsia, a ua pili me ka kiʻekiʻeʻakika;
  • gastroesophageal reflux maʻi (symptomatic);
  • Zollinger-Ellison maʻi pale.

Contraindications

E hoomakaukau ai "Losek CI" hiki ole ke hoakaka ia no ka hypersensitivity ka hoʻomanawanuiʻana i ka omeprazole like maikai i hookomoia benzimidazoles 'ole' ē nā mea hoʻohui i nā hapa o ka lāʻau.

Ua E hoi e kaulana ia ua hoakaka ia keia k me ka mālama nui i loko o ke alo o kanaka na hiʻona me noho'na makaainana i ulu kaumaha poho, dysphagia, pinepine ka luaʻi a me ka luaʻi o ke koko. Eia kekahi, ma ka gastric ulcer ( 'ole kēia maʻi) e hookaawale ia i ke alo o ka malignantʻeho. O ke kumu ho i ka mea e iapaau ana me ka omeprazole hiki wale makakiʻi na symptoms, aʻauʻa i ka pololeiʻike.

Pehea e lawe i ka lapaau "Losek CI" (20 mg)?

O na dala e wale e lawe hōʻike waha 'i loko o ke kakahiaka. Ka lāʻau 'E e aleia a pau, me ka wai. Ka lāʻau 'E i paopao ai nau.

Nā papa e ae, e hoike mai i loko o ikiʻakika kinowai a me ka wai (e laʻa me, ma ka hua Piʻihonua). Naʻe, ka mea kūpono pāʻoihana e e hoʻopauʻia i loko o ka hora.

I ka esophageal reflux, gastric a duodenal ulcer he 12-makaukau ana ua hoakaka ia 20 mg kekahi manawa i ka lā. I ka reflux esophagitis mahele lāʻau mahuahua i nā manawaʻelua.

Ka lōʻihi like 'ole o ka iapaau ana o ka ulcer no 2-4 pule ma reflux esophagitis - 4 pule, a me ka gastroesophageal reflux - 4-8 pule. E pale aku relapses o ulcers a me reflux oesophagitis i o ka lanakila i ka hou o ka loaa ana i ka lāʻau i loko o ka mahele lāʻau o 10 mg.

ʻaoʻao waiwai

Medicine "Losek CI" analogs lāʻau paha iʻaoʻao loa. Ka loa, he pono ole i na kēia pathological keia: headache, flatulence, abdominalʻeha, constipation, diarrhea, nausea a me ka luaʻi.

No ka infrequentʻaoʻao 'ole nā dermatitis, hives, pōniuniu, ka ohane, paresthesia, poʻe noʻonoʻoʻole, malaise, drowsiness, a piʻi aʻela ka haʻawina o ke ake nā'ūhū, a me ka Kanikani'āʻula.

Aho pohihihi keia i loko o nā mea maʻi loaa omeprazole ai ka haohao ana hypersensitivity reactions (e laʻa me, anaphylactic kŰia, kuni, anaphylaxis, angioneurotic edema), a me ka bronchospasm, hepatitis, Muscle nawaliwali, hepatic e hemahema, leukopenia, encephalopathy, arthralgia, kaumaha, myalgia, pancytopenia, thrombocytopenia, manaʻo pīhoihoi, agranulocytosis, maloo waha, hyponatremia, gastrointestinal candidiasis, aggression, photosensitivity, ka huikau a me ka blurred hihiʻo, hallucinations, sweating, ono haunaele, Periph -geometric edema, stomatitis, interstitial nephritis, alopecia, gynecomastia, erythema multiforme, microscopic colitis, Stevens-Johnson maʻi pale a me kaʻawahia epidermal necrolysis.

Loa kākaʻikahi malama hypocalcemia, hypomagnesemia, hypokalemia a me ka hypomagnesemia.

Medicine "Losek CI": uku a me analogues

Ke hoʻohālikelike i like ai ', i ke kumukuai o na dala mea he kiʻekiʻe. No laila, no ka 14 papa oe, e loaʻa, e uku ma kahi o 250 Lūkini rubles. Noonoo pono i ka lōʻihi makahiki hooponopono o ka medicament (2 i 8 pule), i ka iapaau ana i kekahi pipiʻi no ia.

Ke pani no ka lāʻau "Losek CI"? Analogs o ka mea paahana i ka ia ka hoʻokōʻana. Naʻe, ma mua ana ia, eʻoiaʻiʻo, e kukakuka pu me kou kauka.

No laila, e puku i ka lapaʻau "Losek CI" e ia i ka i kēia lapaʻauʻia: "Omeprazole'Acere", "Vero omeprazole", "Tsisagast", "Gastrozol", "Helol", "Demeprazol", "Helitsid", "Zhelkizol", "Ultop "" Zerotsid "," Ulkozol "," Zolser "," Ulzol "," Krismel, "" ka Soprano, "" Losek "," Romesek "," Omez "," Promez "," Omez D "," Pleom- 20 "," Omez Insta "," Peptikum "," Omezol "," Otsid "," Omekaps "," Ortanol "" Omeprazole "" Omitoks "" Omeprazole Richter, "" Omipiks "" Omeprazole STADA " "Omizak", "Omeprazole Zentiva", "Omefez", "Sandoz Omeprazole", "Omeprus", "Omeprazole-OBL", "Omeprazole-FPO" "Omeprazol-Teva", "Omeprazole-Ako".

e hoike

He aha nā mea maʻi i aku nei au e pili ana i ka lāʻau "Losek CI"? Comments e pili ana i keia hale, he mau'āina maikaʻi. E like me ka poe i loa ua olelo mai medicament, ka mea, ua hala loa ka pono e lawe aku oe i na symptoms o kaʻakika o gastric wai. A me ka hopena o kekahi 'kokoke koke ma hope o' ai, inu o ka papa (1-2 hola).

Pinepine noʻonoʻo i nā mea hoʻohana i heartburn a me he ahi ka waiʻona ma ke kua o ka breastbone.

I loko nō o ka ka hoʻokōʻana kiʻekiʻe o ka lāʻau, loa nā mea maʻi ohumu ia ma hope o ka hoopau ana o kona komo discomfort hoi aku la. Ma keia hihia, kauka waiho aku i ka hoʻomaka i ka hulina lapaau a me ka lapaʻauʻia ana ma ka liʻiliʻi eha pule.

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