'O ka ma'iNā Hana

Nā Analogues a me nā'ōlelo a'o no ka ho'ohana'ana i "Lomefloxacin"

He aha ka mea e hiki ke pani i kahi huahana lā'au e like me Lomefloxacin? 'O nā analogs o kēia lā'au lapa'au,'o kona kumu, nā mea'alohia e ho'ohana ai a me nā pono kīwila e kama'ilio'ia ma lalo nei. Eia kekahi, e a'o'oe pehea e ho'ohana pono ai i kēia mea hana, a me ke'ano o nā mea hana.

'O ke'ano o nā lā'au lapa'au, a me kona hō'ailona

I loko o ka pahu hea ka mea i hana'ia? 'Auhea kahi a'o e ho'ohana ai? "Lomefloxacin" he papa i ho'onohonoho'ia i loko o nā pu'u a ho'opa'a'ia i nā paila pepa me ka hō'ike.

He aha nā mea'ai o ka huahana? 'O ka mea hana o kēia lā'au lapa'au'o Lomefloxacin hydrochloride. Ho'ohui pū'ia kekahi mau papa hana kōkua.

Nā hua lā'au lapa'au o ka lā'au lapa'au

He aha nā papa Lomefloxacin? Ke'ōlelo nei ke kumu he huapona bactericidal antimicrobial e pili ana i kahi hui o nā lā'au'alopelohe,'o ia ho'i, fluoroquinolones, a me ke'ano o ka lua o nā hanauna o kēia mau lā'au lapa'au.

He aha ka mea e ho'oholo ai i ka maika'i o ka lā'au antimicrobial o ka lā'au i noi'ia? Ua loa'a kēia mau mea o ka papa Lomefloxacin (400 mg) ma muli o ka mea hiki i kāna mea hana ke hiki ke ho'oikaika i kahi hopena o ka DNA-gyrase ('o ia ho'i ka enzyme bacteria), e ho'olako i ka pū'ulu. Eia hou, ua hana kēia luna i kahi pūnaewele pa'a (complex) me kona tetramer, a ke luku nei ho'i i ka palapala a me ka ho'opi'i'ana o ka DNA o nā pūpū bacteri, a'o ia ke kumu o ka make'ana o lākou.

Hō'ike'ia ka hana i hō'ike'ia o kēia lā'au me ka nānā'ana i kēlā'ano bacteri'aiapika maika'i e like me gonococcus, salmonella, pseudomonas aeruginosa, hemophilic a me ke kōpū o ke kino, ka mea hana causal cholera, meningococcus, shigella, morganella a pēlā aku. Eia nō ho'i,'o ka lā'au "Lomefloxacin" (400 mg) ka hopena kaumaha ma luna o nā proteins, chlamydia, campylobacter, mycoplasma, legionella, some pneumococci and staphylococci.

Mākou hiki ole ke olelo i ka olelo mai lāʻau mea nui mana e ku e Mycobacterium tuberculosis. Hiki iā ia ke ho'ēmi i ka manawa o ko lākou hopena, a me ka ho'onā wikiwiki loa o ka ho'opuka'ana.

Ke mālama'ia ka hopena maika'i o Lomefloxacin me kona mau li'ili'i li'ili'i i ke koko. Inā keia ia'ku ua malama loa kākaʻikahi.

'O ka ikaika o nā lā'au lā'au

Pehea e ho'omo'a'ia ai nā lā'au? He aha ka'ōlelo a'o e ho'ohana ai? Lomefloxacin kahi mana ho'ona'auao maika'i. Ma hope o ke kau'ana i ka lā'au lapa'au, hiki i ka hō'ailona plasma ka lō'ihi i 55-55 mau minuke.

Me nā pāpona plasma,'o kēia lā'au lapa'au wale nō ia e 10% wale nō. He mau'ano ho'ona'auao maika'i ho'i ia i nā'ano a me nā mea like'ole (e like me ka genitalia, nā hui, nā'ōpū o ka'ōpū, nā pūnoa ENT, nā'ano pelvic, iwi, peritoneum, nā mea lewa, a me nā mea'ē a'e), kahi o kona helu he 5-7 manawa ki'eki'e. Plasma.

Pono e ho'omaopopo'ia ua ho'okomo'ia kekahi o ka lomefloxacin a ua hana'ia kekahi mau huahana.

'O ka manawa ho'omaha o kēia lā'au lā'au he 9 mau hola. Ho'opuka'ia i loko o ka ho'opili'ana me ka urine (70-85%) a me nā feces (25-30%).

Nā kuhikuhi no ka kuhikuhi

'Ai nā kānaka i'ike, akā i loko o ka'umehana kālepa hiki'ole iā'oe ke loa'a nā palapala Lomefloxacin wale nō, akā'o Lomefloxacin + Pyrazinamide + Prothionamide + Etambutol + Pyridoxine. I kēia hihia, ua hō'ike'ia nā lā'au i'ōlelo'ia'elua no ka ho'ohana'ana inā:

  • Nā ma'i'ele'ele o ka'ili, a me nā mea'olu'olu (e like me nā ahi, nā'eha i ho'opō'ia, a me nā mea'ē a'e);
  • Osteomyelitis;
  • 'O Chlamydia a me gonorrhea (e like me ka bloodpharoconjunctivitis a me ka chlamydial conjunctivitis);
  • Nā'eha o ka'ōhula pahū (e like me ke cholera, ka ma'i dysentery, ka ma'i typhoid, salmonellosis);
  • Nā ma'i'eha o ka hanu (e like me nā hanana'ana o ka ma'i hānai ma'i);
  • Nā pō'ino o nā alalele bile;
  • 'O nā ma'i i loko o ke kikowaena holoholona (e like me ke'ano o ka ma'ihuta, prostatitis, cystitis, pyelonephritis);
  • 'O ka ma'i o ka'ōpiopio (e like me ka ho'oponopono'ana o nā kānaka me ka holomua o nā ma'i o ka ma'i, a me ka pi'i'ana i ke isoniazid a me ka rifampicin a me ke kū'ē'ana i ka chemotherapy);
  • Ma mua a ma hope o ke kāpili'ana o ke transurethral (no nā kumu hana wale nō).

Ho'oku'u'ia e kau i nā palapala antimicrobial

I nā nīnau hea hiki'ole iā'oe ke ho'ohana i nā lā'au lapa'au i nīnau'ia? He aha ka mea e ha'i mai nei iā mākou e pili ana i nā kuhikuhi no ka ho'ohana'ana? Ho'opi'i'ia'o Lomefloxacin no ka ho'ohana'ana inā:

  • Ke lawe'ana i ka'ōpū;
  • Ka hānai'ana;
  • Ka'ike pilikino o nā mea'ai o ka hui o fluoroquinolones;
  • I ke kahi li'ili'i (hiki ke hana i ka pale'ana i ka ulu'ana o ka pūpū).

Nā kuhikuhi no ka ho'ohana

"Lomefloxacin" - nā papa, i hō'ike'ia wale i ka ho'oponopono waha. Pono lākou e lawe ho'okahi i ka lā, no ka'ai'ana, e inu ana i ka 230 ml o ka wai ma'amau.

'O ka lō'ihi o ke kau'ana me kēia lā'au lapa'au ma luna o ka hō'ailona, a me ka pa'akikī o nā ma'i a me ke'ano o ka ma'i.

'O ka ma'i bronchitis a me ka bronchopneumonia o ka papa'auhea e mālama'ia me kahi lā'au like 400 mg o ke lā'au no nā lā he'umi.

I ka mālama'ana i ka chlamydia (urogenital), me nā ma'i bacterial chlamydia a me gonorrhea-chlamydial, ua ho'onohonoho'ia nā ma'i i 400-600 mg o lā'au lā'au i kēlā lā i kēia lā, me ka lō'ihi o nā lā he 28.

Ho'oma'a'ia i nā hanana'ana o ka'ōneumonia pa'akikī a me ka bronchitis o kahi'ano ma'amau e ho'okō'ia i nā hana o nā lā a pau me 400-800 mg o ka mea kono no'elua pule.

I ka mycoplasma maʻiʻaʻai manaoia lāʻau hoakaka i 400-800 mg no ka lā, a me ka lōʻihi o ka hooponopono ana o na papa i loko o 3 pule.

Hiki ke mālama'ia nā ma'i ma'i o ka'ōmumu e 400 mg o ke lā'au lā'au. I kēia hihia, mālama'ia ka mālama'ana i nā hihia hihia'ole no 5 mau lā, a ua pa'akikī - 14 mau lā.

Me ka gonorrhea o kahi'ano'ano nui, ua'ōlelo'ia ka lā'au "Lomefloxacin" no ka lawe'ana i kahi'ano 600 mg. No ka ma'i ma'amau o kēia ma'i, ua mālama'ia ka mālama'ana me ka pilikino li'ili'i. I kēia hihia, ua lawe'ia ka lā'au i loko o kēlā me kēia lā no 5 mau lā.

'O ka hō'ailona o ka ma'i'ōma'oma'o e hiki ke lawe i nā lā he 14-30 (i kekahi manawa a hiki i nā mahina 3). Ho'oma'i'ia kēia ma'i i 200 mg mau manawa i ka lā.

I loko o nā ma'i hō'ailona o ke'ano ko'iko'i a i'ole ke'ano, a me ka po'e e halihali ana i ka hemodialysis, ua'ōlelo'ia'o "Lomefloxacin" i ka nui o 400 mg i ka lā, me kona ho'onui'ana i 200 mg.

Phenomene o kahi'ano maika'i'ole

He aha nā hopena maika'i'ole o nā papa Lomefloxacin? Ke kuhikuhi nei ke kuhikuhi i kēia mau kuhi:

  • 'O Bronchospasm, ho'onui i ka ho'ohemo'ana o ka'ōpū, kausea, ka'ī, dysphagia;
  • 'O Dyspena, lua'i, nā ma'i o ka'ōpū, ka diarrhea, dysbiosis;
  • Nā hō'ailona like'ole, ke'oki i ke kīpē, ke'eha epigastric, ke kīpona;
  • 'O ka nui o nā ki'eki'e o nā enzymes o nā mo'o,'o ke kaha malo'o, ka GIT kahe'ana;
  • Ka ho'omau'ana, ka hō'ailona'ana, ka palekana bipi, ka wehewehe'ana i ke alelo, myalgia;
  • pseudomembranous colitis, headaches, loli ma ka ikaika loa ka makemake, vasculitis, pōniuniu;
  • 'O ka'ōnēnia, ka eha o ka pahu a me ke kua, ka asthenia, ka maka'u'ole, ka mana'o o ka malaise general, ka pu'uwai, ka ha'alulu;
  • 'O ka Hyperkinesis, ka luhi luhi, nā ha'alulu, nā hana;
  • 'O ka'eha i nā maka, ka wala'au a me ka'eha i loko o nā pepeiao;
  • 'O Dysuria, ka ho'onui'ana i ka hau'oli, ka hematuria, ke kuhihewa;
  • 'O Crystaluria,'ike'ole;
  • Albuminuria, glomerulonephritis, leukorrhea, edema, polyuria, epididymitis, pa'akikī urinating, orchitis, pāohana kaumaha;
  • Cyanosis, anuria, hypotension, vaginitis, tachycardia, extrasystole,'eha peineineal, bradycardia;
  • intermenstrual kahe ana ke koko, thrombocytopenia, vaginal candidiasis, myocardial infarction, cardiomyopathy, phlebitis;
  • Ka pi'i'ana o ka ma'i'ole a me ka stenocardia, ka'oihana purpura, ka ma'i kalapili, ka'ili'ana o ka'ili;
  • Ho'olālā pā'ani, ki'i ki'i, ha'awina fibrinolysis nui, urticaria, lymphadenopathy, hyperhidrosis;
  • Kahe'ana o ka Nasal, ka erythema keu (ka'ākau), ke'ano o ke kani, ke kī, ka wela;
  • 'O ka Superinfection, ka hypoglycemia, ka makemake, ka make wai.

Ho'opau'ia me nā hua'ōlelo

I ka hihia o ka loke o Lomefloxacin, ua'ike nā ma'i i ka nausea, nā'epa erosive o ka mucosa'ōpū, ka lō'ihi o ka wā QT, nā mana'o nui, ka ho'onāukiuki, ka hilahila, a me ka pi'i'ana i nā hā'ina kūpono.

I ka'ike'ana i ke kūpono'ole o ka hemodialysis i ke'ano o ka ho'olō'ihi'ana,'o ka hopena o nā kūlana i luna nei e kau'ia ma luna o nā hō'ailona o ka loa'a.

'O ka pilina me nā lā'au'ē a'e

Ke hui pū'ia'o Lomefloxacin me Teofillin, ua aneane hiki'ole ke kāohi'ia kona pili.

A hiki i ka wā hoʻokahi aaieieno? O antacids a me sucralfate e hana chelate eiiieaenu i emi ai ka bioavailability o lomefloxacin. 'O ke kumu ke kumu o ka lō'ihi ma waena o ka lawe'ana i kēia mau lā'au i 4 mau hola.

'O ka ho'ohui pū'ana o "Lomefloxacin" a me nā ko'i nui o ka mea kalo e ho'onui i ka hapalua o ka hopena.

I ka wā e hana ai i ke kīkoko, mai lawe i ka lā'au lapa'au me ka "Rifampicin", i'ole e alaka'i ia i ke antagonism o ka hana.

Hiki i nā ho'olaha like'ole o nā NSAID ke ho'onui i ka hō'ino o nā lā'au lapa'au a hiki ke ho'oku'u i ka hopu.

"E hiki i ka Lomefloxacin ke ho'onui i ka maika'i o nā mea hana'ele'ele kūpono no ka ho'oponopono waha.

'O nā lā'au,'o ia nā'āpena o ka ho'opalele'ana o ka pulupili, e kāohi i ka excretion o "Lomefloxacin."

Nā Kūkākūkā Kūikawā

I loko o nā hō'ailona ma'amau, pono ka ho'onā'ana o ka hō'ailona pono, e hilina'i ana i nā ho'ohālike QC.

No ka lō'ihi o ka ho'olālā, pono pono ke kāohi i ka ho'olā'ihi lō'ihi i kekahi mau kumu o ka ho'ouluwe uila ultraviolet, me ka lā o ka lā.

Ho'olako'ia nā mea'enela lā'au, me nā pāpili'ene mineral, 120 mau minuke ma mua o'ole ma mua o ka lawe'ana i nā papa i nīnau'ia.

'O nā lā'au like'ole

'O ka lā'au lā'au "Lomefloxacin" he nui kona mau ana. Ho'omaopopo nā kānaka'ike i nā mea hou no nā kumu nui: Abaktal, Elefloks, Zanotsin, Tsifran, Avelox, Tsiprolet, Zofloks, Cyprinol, Quintor, Ciprofloxacin, Levofloxacin "," Lehuaflox ","'Oloxacin "," Norbaktin "," Ofloks "," Norfloxacin ".

Nā papa Lomefloxacin: hō'ike

Me ka pūnaewele kūpa'a o kahi hui hānai e pili ana i ka lua o nā hanauna o ka fluoroquinolones, a me ke koho pololei'ana i nā lā'au lā'au a me nā lā'au ho'omalu lō'ihi,'o ka ho'olālā e pili ana i ka luna i nīnau'ia he'ano maika'i loa.

Wahi a nā pane o nā mea ma'i, ua hō'oia kēia lā'au'ai he lā'au lapa'au maika'i e pili ana i nā'ano microinganu. Eia na'e,'ōlelo kekahi po'e'ōlelo i kekahi manawa ua ulu kēia lā'au i ka ho'oulu'ana o kekahi mau hopena, akā, ma ke'ano he kaulike,'ōlelo mālie'ia a hele'ole paha lākou ma hope koke iho o ka hopena o ka ho'okolohua.

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