Ola kino, Hoomakaukau
"Ortanol": mea kōkua, aʻo no ka hoʻohana 'ana, maoli
He aha mea i ka lāʻau "Ortanol"? Mai mea kōkua i ka laau? Nā pane i kēia mau nīnau hiki ke loaʻa ma lalo nei. Eia hou, ke haawi i ke kumukuai o ka olelo mai huahana, kona contraindications, analogs a hoʻokuʻu ano.
'ōpala i ka lāʻau, kona haku mele 'ana, hōʻikeʻano, ano
E hoomakaukau ai "Ortanol" ua i loko o ka palapala o ka paakiki capsules nui № № 1 ole 2. kēia 'o ia hoʻi, he keʻokeʻoʻeleʻele, e like me ka palapala «OME 20» a «OME 40' (ke kaumaha ma muli laʻau heluna). Maʻiʻo lāʻau lapaʻau capsules ho i ka hulu pellets.
E nā ka lapaʻauʻia "Ortanol"? Reviews paipai i na kumu o ka waiwai ua noʻonoʻo pono i ka lāʻau omeprazole. Nō hoʻi ka mea, he kākoʻo eiiiiiaiou e like me croscarmellose paʻakai, haʻahaʻa hookomoia giproloza, lactose anhydrous, microcrystalline kelulose, hypromellose phthalate, povidone, polysorbate 80, talc a me ka dibutyl sebacate.
I ka haku mele 'ana o ka mea hōʻikeʻikeʻuʻuku iwi nā: propylene glycol, hypromellose, butanol, carrageenan, anhydrous ethanol, shellac, potasiuma koloriside, anhydrous isopropanol, titanium'okikene lua, ka inika no kakauia a me ka wai.
I kuai medicament "Ortanol" (mea hōʻikeʻikeʻuʻuku) komo i ka blister, pūʻolo helu i ka pepa pahu.
Pharmacological hana o ka lāʻau
He aha mea he "Ortanol" (mai ka mea kōkua kēia lapaau, oe e aʻo lalo)? E like me na kuhikuhi, me ka lāʻau o ka inhibitor o proton EII ni. Ua ho'ēmi i kāʻakika-i? Iecaianoaaiiuo, 'o ia hoʻi,' aʻole hoʻi ia i ka ha awina o K + -h + -ATPase i loko o ka opu, a he oiaio, ua i loko o kona parietal keena. Nō hoʻi ka mea, ālai 'ke kahua hope loa o gastricʻakika secretion.
Uluwehi O "Ortanol", ke kumukuai o ka i ua helu 'ia ma lalo iho nei, o ka prodrug. Keia mea paahana ua ho'ā 'ia i loko o kaʻakika meakino o na tubules (secretory) parietal keena. Eia hou, e ho'ēmi i kā ka hauma¯na kahi a me ka basal secretion nānā 'ole o ke ano o ka stimulus.
Antisecretory waiwai o ka medicament ana i loko o ka mua 60 minuke (i kā mākou ma hope o 2 hola). Inhibition o 50% o ka i kā mākou secretion mau mawaena o ka lā.
A hookahi mahele lāʻau o ka lāʻau e hoʻolako pono a me ka kokololio suppression o nighttime a me ka ao, gastric secretion. Kona i kā mākou mea hiki i ka 4th lā o ka lapaau, a nalo ma hope o nā lāʻekolu ma hope o lapaau.
Kinetic waiwai o ka ai '
Ma ka loaʻa 'o ka "Ortanol" e hoomakaukau ai ka mea loaʻa iā ia nā kiʻekiʻe omo. Peak nā hoʻohui like o omeprazole i loko o ke koko ma hope o ka malamaia 0.5-3 hola. Ke loa bioavailability o ka lāʻau o 30-40%, a me ka medicament pilina me ka wai koko nā polokina - 95%.
Omeprazole pūnao ma ke akepaʻa, e lilo eono pharmacologically AEeOEXAaI nā mea loaʻa.
Ka hapa-ola ka lapaʻauʻia manawa mea 0.5-1 hola. Ia auoiaea ia e like me nā mea loaʻa ma ka hakuʻala (70-76%) a pu me ka bile (18-24%).
People me ka maʻi akepaa nā maʻi bioavailability o ka lāʻau ua me ka nui loa, a mahuahua nui, a me ka wai koko hapa-ola ihoiho 3 hola.
Ma nā mea maʻi me ka maʻi hakuʻala maʻi excretion 'aʻole hoʻi ia. Kēia ia lŘlŘ i kupono i ka ka ho'ēmiʻana i loko o CC.
Medicament "Ortanol": aha kokua?
Nānā akula au i ko lakou hoomakaukau ana ua hōʻike no ka hoʻohana 'ana i ka mea kēia mau maʻi:
- reflux esophagitis;
- gastrointestinal ulcer maʻi kino (me relapse Kāohi);
- hypersecretory Hawaii (stress ulcers o ka naʻau liʻiliʻi, Zollinger-Ellison maʻi pale, systemic mastocytosis, polyendocrine adenomatosis);
- eradication o Helicobacter pylori iho mailoko o nā mea maʻi me ka ulcerative mai o ka digestive'āpana (ma ka hui pu ana, Inc);
- lapaau a me ka Kāohiʻana o gastrointestinal mucosal poino nā loko i i kena ae la o NSAID (mucosal ka'aʻaiawā, dyspepsia, peptic ulcer).
Bans ka hana ai '
He aha e na contraindications lāʻau i "Ortanol" (mai ka mea i hana i keia mea paahana, ua hai aku ma luna mākou)? E like me na kuhikuhi, noʻonoʻo i ka lāʻau 'hiki ole e hoʻohana' ia:
- lactation;
- i kamaliʻi;
- hypersensitivity i ka lāʻau waiwai.
Me ka kūikawā mālama nui noʻonoʻo lāʻau i hoakaka ia no kaʻaʻa puʻuwai a me ka ake ole.
Uluwehi O "Ortanol": olelo
Kēia lāʻau 'ua kuhikuhi wale maloko. Ua ua ia pono ma mua o kaʻai (i hookuu i ke kakahiaka mua aina kakahiaka).
I ka mea hōʻikeʻikeʻuʻuku a me ka lāʻau e aleia i ka pau i ka wai. Ma ia hihia, ina o ka hoʻomanawanui mea hiki ke hoʻohana i ka lapaʻauʻia loa, kona Contents hiki e ia ka pono i loko o ka uuku dala mea,ʻaʻole loaʻakika wai.
Ke laʻau heluna o ka lāʻau hilinaʻi nui ma luna o ka hoike.
I ka ulcers 12 duodenal ulcer medicament ua lawelawe ma 20 mg koke i ka lā i mau pule. I ka hanana ana ma hope o ka mua makahiki piha scarring 'aʻole i hoʻomaka ai, hou-i'ōleloʻia ai nā-hebedoma Inc.
Ma ulcerative maʻi hoʻopale i ka lapaʻau, i kēia hope paha ua pono, e lawe i ka laʻau heluna o 40 mg koke i ka lā. I ka papa o ka Inc me keia k hiki e hoopomaikai io no eha pule.
Capsules "Ortanol" nāʻikepili a i ua helu 'ia ma luna, ulcerative lesions o ka'ōpū lawe 20 mg koke kela la i keia no eha pule. Inā scarring Aʻole ole ana ma hope o ka hala makahiki, me ka hou-i'ōleloʻia ai, eha-pule Inc. Ma gastric ulcer, hoʻopale i ka lapaʻau, ka lapaʻauʻia ua? Aeiiaiaoaony e lawe i kekahi mahele lāʻau o 40 mg koke i ka lā (i ka uku o ka mai i ewalu pule).
Eradication o Helicobacter pylori ua lawe mai i loko o ka hoʻohui pū Inc. Ma keia hihia, ke medicament ua lawelawe ma 20 mg palua i ka lā ma muaʻai (no elua pule) ma ka hui pu ana, me ka antibacterial konohiki.
I ka reflux esophagitis lāʻau ua? Aeiiaiaoaony e hoʻohana i ka nui o ka 20 mg (hookahi) no eha pule. Inā kēiaʻano hana i ka k mea ole conducive ia ke hoʻokō 'hoolaia, ke hoʻomanawanui ua hoakaka ia i ka lua o ka papa (eha pule). I loa reflux esophagitis lapaʻau keia mea paahana ma ÿö mai i ewalu pule.
I ka hypersecretory moku'āina ua noʻonoʻo i ka lapaau no ka heartburn lawelawe pākahi. Ke paipai hoʻomaka laʻau heluna no nā mākua, he 60 mg (hookahi), a me ka mea i kā mākou - 120 mg.
I kauoha mai ai i ka lāʻau 'oi ma mua o 80 mg no ka lā, ka mea, ua maheleia i loko o kekahi mau kahua o ka hoʻonaʻauao.
I ka gastrointestinal mucosa hui, kēia pōʻino, a i ke kumu e NSAID, e like me ka Kāohiʻana o ka mea hōʻikeʻikeʻuʻuku "Ortanol" waiho aku i ka hoʻohana 'ana o kekahi mahele lāʻau o 20 mg kēlā lā, ma mua aina kakahiaka (no ka mea holoʻokoʻa lōʻihi like' ole o NSAID Inc).
No ka poʻeʻelemākule kanaka a me kanaka me ka loa ake maʻi i kā mākou kela la i keia mahele lāʻau o 20 mg.
No nā mea maʻi me kaʻole hakuʻala papa laʻau heluna hoʻoponopono ua koi 'ia.
ʻike manaʻoʻaoʻao
He aha reactions objectionable ma o na la lāʻau "Ortanol"? Reviews aku nei au i ka i kēiaʻaoʻao ole:
- headache, blurred hihiʻo, pōniuniu, erythema multiforme, paresthesia;
- drowsiness, nausea, ono haunaele, diarrhea, Kanikani'āʻula, flatulence;
- manaʻo pīhoihoi, maloo waha, kaumaha, maʻi, reversible noʻonoʻo hilahila;
- encephalopathy, gynecomastia, hepatitis,ʻike ākea edema, ka luaʻi, a me ka photosensitivity;
- abdominal eha, thrombocytopenia, constipation, pancytopenia, mahuahua o kona'ākilikai phosphatase ha awina, a ake transaminase;
- itchy ili, hoʻopōʻino ake hana, Muscle nawaliwali, i ke kahua o ka gastric glandular cysts;
- alopecia, eosinophilia, mahuahua sweating, bronchospasm, agranulocytosis, angioedema;
- leukopenia, myalgia, kuni, arthralgia, anaphylactoid reactions, urticaria, interstitial nephritis.
ʻaoʻao waiwai e ana i loko o ka noi o ka hōʻike 'ana no konohiki i mehana a me ka transient ma ka ano.
hihia o ka overdose
I ka lawe ana ka lapaʻauʻia no ka heartburn i loko o ka hoomanawanui kēia mau symptoms kānāwai: headache, maloo waha, tachycardia, drowsiness, nausea, blurred hihiʻo, ka luaʻi, ka hilahila, mahuahua sweating.
Ma lalo o ia mau rula, symptomatic Inc.
lāʻau hana kūleʻa
Together me ke komo omeprazole mahuahua hapa-ola, a mahuahua lehulehu "Diazepam", "warfarin", "phenytoin", e like me 'ē ai' i i metabolized ma ke akepaʻa, me ka isoenzyme CYP2C19.
Omo ano hiki ke nee, ka bioavailability o ka i me ka nānā 'ana i kaʻakika o gastric wai (e laʻa me, "Itraconazole" "ketoconazole" nā mea kemika o ampicillin "cyanocobalamin" a me ka hao paʻakai).
Ke bioavailability o digoxin ka wā ke kākoʻo '-lawelawe me ka omeprazole ua hoomahuahua ia ka 10%.
Nānā akula au i ka lāʻau 'hoʻokāʻoi aʻe ana i ka inhibitory ia ma ka'ōnaehana'ē aʻe hematopoietic ai'.
No clinically nui lāʻau hana kūleʻa me antacid ai ', caffeine, "theophylline", "Quinidine", "propranolol", ethanol, lidocaine a "metoprolol" ua i kau.
kekahi koi
malignancy E e hoʻokoe 'mua hoʻomaka kanaka me ka omeprazole. O ke kumu ho i ka mea i keia k Inc ke makakiʻi na symptoms, aʻauʻa i ka pololeiʻike, hoakaka.
Currently, eiaʻaʻoheʻikepili ma o ka hopena o na dala ma ke kanaka ka hana i ka pāʻana maomeka, a kipaku kaa.
Kāki a me analogues
Pehea ka nui o kēia Anati-ulcer lāʻau ', like "Ortanol"? Ke kumukuai o keia k mea e pili ana i 100-115 rubles. No ka hapanui o nā mea kūʻai mai, i ka lilo ana o keia, ua maikaʻi nō.
He aha e puku i ka lāʻau "Ortanol"? Analogs o keia la hoomalolo e hōʻike mai iā ia i loko o ka palapala o ka "omez", "Loseprazol", "Gaseka", "Omelika", "omeprazole".
Reviews
Reviews o capsules "Ortanol" mea maikaʻi i ka oi loa. Nā mea maʻi i aku nei au i ka lāʻau o ka hoʻokō antiulcer hope paha. Ua koke eliminates heartburn, a me ka manao ana o kaʻehaʻeha, a kuni i loko o ka'ōpū.
Kilo'ōlelo aku nei au i ka lāʻau ma ka ninau mai i ka maikaʻi ia ma luna o ka papa o ka maʻi o ka digestive'āpana wale ina kona? Eaia, ua hoonohoia ma ka gastroenterologist. Kauka hōʻike i kā lākou iho, e lawe i kēia k ua hookapuia, e like me ka mea i he nui loa ikaika ia.
Aia Ua hoi he maikaʻiʻaoʻao o kēia ka lapaʻauʻia nā kona loaʻa nui a me ka haahaa kāki.
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