Ola kino, Hoomakaukau
"Theophylline": olelo ao no ka hoʻohana. "Theophylline": nāʻikepili no ka hoʻohana ana i analogues
Inā poino kekahi kanaka mai ka airway iaʻi, i kēia e hōʻike i ke alo o ka maʻi obstructive pulmonary maʻi (COPD). Kēia maʻi i hala loa, he pono ole. Pinepine i ka hanana o kēia maʻi ike i ka paka. Ka hooulu ana o keia maʻi ua kena aku ma ka maʻiʻaʻai LIKE, a me nā mea kekahi akemāmā ka pōʻino. A kanaka me ka airway constriction hiki apuepue Exhale.
hōʻikeʻano
"Theophylline", kona haku mele 'ana e ho'ākāka' ia ma lalo e, o he keʻokeʻo mea pōaka ka pauka. He iki wailana i ka wai huihui (i loko o ka lākiō 1: 180), akā, ua hikiwawe mea hoʻoheheʻe i ka wela o ka wai (i loko o ka lākiō o ka 1:85). Ua i hoike mai i ka alkalis a me nāʻakika.
'ole
Ma keia hoʻomanaʻo i ka papa kuhikuhiEʻeleu 'Oponopono mea theophylline. ʻaneʻi nō hoʻi nā kekahi kākoʻo eiiiiiaiou. O - lactose monohydrate, makanekiuma stearate, talc, methacrylicʻakika.
hookuu palapala
Aia i mau laha 'ma keia pili ana. "Theophylline" ua hanaʻia e like me ka malama aku-hoʻokuʻu papa (0.1 g., 0,25 g), capsules (0.125 g., 0.5 g), a me nā suppositories (0.2 g).
pharmacological hana
Functionality o ka la hoʻomanaʻo mea nunui-faceted. "Theophylline", hōʻike manaʻo o ka mea e 'oluʻolu, hoʻomaha i hana nāʻiʻo o ka bronchi, ua i ka noho haumāna kahi a me ka vasodilator hana. Kēia makaukau e hōʻoiaʻiʻo ka maʻamau hana o ka naehana waena. Hoʻopau ka eha ma ka diaphragm, a hoʻoikaika i ka functioning o ka intercostal nāʻiʻo i ka poʻea pau e "Theophylline". Kona hoʻohana ma o ka maʻamau kaʻina hana ho'ēmi i kā ka pahiki o ka hoike ana mai o allergic reactions i loko o ka naehana'ōnaehana type kino. I aku la ko lakou hoomakaukau ana ke kulia i ka diuretic hopena. Ke alo aku o ka hana 'ona i loko o ka medicament ka paipai' ana i ka normalization o naehana papa, hoemi i ka nui o ke kalapona'okikene lua, a mahuahua hoʻokomo ea.
nāʻikepili
E hoʻomana aku la lāʻau ma hanana o bronchial asthma, asthmatic kūlana haʻahaʻa, obstructive bronchitis, pulmonary emphysema. Nō hoʻi ka mea, ua hoʻohana 'ia e like me he kökua i keiki na kamalii uuku me ka apnea. E hoʻohana i "Theophylline" kuhikuhi me ka bronchodilator.
Piha hōʻike o ka pae o ka olelo mai hoʻomanaʻo
Initially, ma ka iapaau ana o ka COPD mea paha bronchodilators. Ka mea, e lawe 'ana Air. I kekahi o kēia mau ai ', e like me ka ua i haiia ae maluna, oia hoomalolo mea like "theophylline". Na Ke Kumu no ka hoʻohana characterizes mea like me ka bronchodilator lāʻau, a hāpai mai i ka ai-i kapaia wahi o ka purine receptors. Ke alo o ia ka hopenaʻano papa hana e hōʻoiaʻiʻo i ka wehe 'ana o spasms i loko o ka'ōlohelohe Muscle o na bronchi, ka hoʻopau o ka eha i loko o ka diaphragm, ho'ā hope o ka o oxygen i na maʻiʻaʻai, ka hoʻomaikaʻi i ka hana o ka intercostal nāʻiʻo. E like me ka hopena, i ka Hawaiian Airlines wehe i, i ke kanaka hanu aho.
Ua loaʻa he definite pono, "Theophylline". Na Ke Kumu no ka hoʻohana i ka 'i keia k hiki ikaika hopena ole wale ma luna o ka ÷ naehana hanu'āpana, akā, no hoi ma nā kino nenoai. Kēia lāʻau kōkua, e hoʻonui i ka ipu coronary a me kaʻike ākea koko, alalai mai i ke kaʻina hana o ka platelet mea pīlali, mea he mehana diuretic hana. Ua i nā stimulation pahi hope o ka naau Muscle (myocardium), haʻahaʻa ke koko, e like me ka pono me ka pono ia ma luna o ka Central ko mākou hopohopo nenoaiu. E like me ka hopena, i ka lāʻau mea hiki ke hana versatile, ka poʻe me antiasthmatic, bronchodilator, diuretic, spasmolytic, vasodilatory a me cardiotonic waiwai.
"Theophylline": kauoha no ka hoʻohana
E hoʻoholo i ka laʻau heluna, he nui na ana hoʻohālike. "Theophylline", e like me ke kauoha, e pono e lawe i ke keiki a hiki i ka makahiki o ka 14 a me nā mākua, 300 mg no ka lā 2-3 manawa. Ma keia hihia, no ka lapaʻau e inu i ka wai i loko o nui mea. Inā pono, hiki e mahuahua ai ka mahele lāʻau a hiki i 500 mg 2 manawa i ka lā, ina e waiho ma kou kauka. Inā i ka hoʻomanawanui i ke kino kaumaha emi o 60 kg, ka laʻau heluna e e 100 mg 2 manawa i ka lā. Ma keia hihia, ka mea i'ōleloʻia ai kakahiaka a me ke ahiahi? Eaia o keia hoʻomākaukau like "Theophylline". Instruction hākālia nō i hoolaia mea pono e hoʻomaka me ka poe liilii, nā māhele a me ke kiʻekiʻe o hoonui ia e ia.
Lālau aʻela ia i ka lāʻau i hāpai keiki, a breastfeeding
"Theophylline" kanawai ma ka fetus ma lalo o ka waeʻano "C" ma ka FDA. Ke hoʻopololei komo iloko o ka placental ke'ākeʻakeʻa mai. Hapai na wahine hiki e mai la lāʻau wale i ka hihia ma kahi pono i ka manao i ka makuahine, ua oi aku ia mamua o ka Loaʻaʻia kamepiula a hiki i ka fetus. I ka wā o ka au trimester a me ka hope o ka pule hāpai keiki e lawe i ka lāʻau, ka malama ana o ka ikaika o nāʻikepili. He nui ke hoomanao.
No ka mea he nui loina paipai i ua hoemi theophyllineʻae i ka III trimester o ka hāpai keiki. Kēia e koi hou pinepine hoʻoholo o ka lehulehu o ka waiwai i loko o ke koko, a me ka hiki ka ho'ēmiʻana o ka mahele lāʻau.
Breastfeeding "Theophylline" hina i loko o ka waiu a me ka hiki i symptoms o irritability i na kamalii uuku a me na hana mana e o kaʻawahia. He nui ka ike. Ka lehulehu o ka la waiwai i loko o ka umauma o ka waiu o ka hola like i kona maʻiʻo ma ke koko lāʻau lapaʻau o ka makuwahine. Nō hoʻi, i kēia 'o ia hoʻi me ka nui loa inhibits uterine contractions.
Contraindications
"Theophylline" kauoha no ka hoʻohana like i ho'ākāka 'ia ma luna, ua contraindicated ina he mea:
- Idiosyncrasy.
- Hyperthyroidism.
- Huʻi myocardial infarction.
- Subaortic stenosis. Kēia mea he pili-hoʻoʻino mai o ka ventricle hema o ka naau Muscle'aʻaʻa. Ua Ua wehewehe aku ma ka olelo o kekahi pahikaua hou o kona lua.
- Arrythmia.
- Epilepsy a me nā convulsive ana.
- Hāpai keiki.
Me ka mālama ia mea e pono ke hana i ka? Eaia o ka lāʻau i ka hoike ana mai o ulcerative mai o ka opu a me ka duodenum.
kekahi koi a
Puhi paka me ka nui loa e loli ai i ke ana o ka pūnao a me ka excretion o na waiwai e like me theophylline. Ua hoʻomanaʻoʻia ai ia. Mea paka 1-2 he huihui 'ana o ka pakalōlō i ka lā, i ka ho'ēmi i kā hapa-ola wā. Ma nā mea maʻi me ka hepatic, cardiac a naehana hoʻokō 'ole' i olelo ia, e like me nā mea palahēhē mea hoʻomaʻi a me hyperthermia ia lŘlŘ deceleration hoʻopau o kaʻeleu waiwai. ? Eaia o ka waiʻona, a caffeine-type huahana hoi mai he nui ia ma luna o ka pūnao o theophylline.
AaOIeIOUIeXAOAaIN
Ka lāʻau "Theophylline" ka paipai 'ana i ka potentiation kanawai o ka β2-agonists. Ua hiki no hoi ka hōʻoi 'tremor, a ua kauoha ia e ka sympathomimetic lāʻauʻano a me ka mea hiki ke inhibit i ke kaʻina hana o ke omo o ka phenytoin. Kali hoʻopau o ka mea ia lŘlŘ i loko o kona AaOIeIOUIeXAOAaIN me ka "erythromycin" a me "phenobarbital." O ia hoʻi, "Theophylline" hoʻolako ka hua i loko o kaʻaʻa puʻuwai excretion o likiuma. Ma keia hihia, i ka pākōlea koena ua pīhoihoi ihola i loko o nā mea maʻi i mea e lawe i ka like paʻakai. Ka lāʻau "cimetidine" ka poʻea pau i ka lehulehu i loko o ke koko theophylline pae, a maoli he i ka manawa o kona withdrawal. Na laau me ka like 'ole, e e helu' ia ma lalo nei.
Ke alo aku o kaʻaoʻao loa
I ka loaa ana o ka olelo mai ai 'ke i kekahi io symptoms. oia:
- Oe e 'ike symptoms o ka pōniuniu, Kanikani'āʻula, headache, maʻule hou ihola nō, uunu nui, tremor, ka hilahila, epilepsy.
- Ma ka mea'ōnaehana mānowai koko'ōnaehana - arrhythmia, tachycardia, wahaheʻe angina, koke emi i loko o ke koko,, angina pectoris.
- Mai ka digestive'ōnaehana - ka muli o nausea, ka luaʻi, heartburn, diarrhea, flatulence, colitis, gastritis.
- A hiki aku i ka hana o ka? Eaia mea hiki e malama kekahi hoikeana o allergic reactions i loko o ka palapala o ka ohane, kuni, urticaria, dermatitis, kuni, sweating a me ka ili rashes.
overdose
Ma keia hihia, eia kekahi mau symptoms. Ma lalo o kēia mau hoikeana Komo:
- manaʻo pīhoihoi;
- hilahila;
- convulsions;
- tachycardia;
- arrhythmia;
- hypotension;
- nausea;
- diarrhea;
- ka luaʻi me ka admixture o ke koko;
- hyperglycemia;
- metabolic acidosis.
A pau kēia mau symptoms ua ia i kekahi kanaka. ʻo ia, lawe mai ma:
- Ho'ā 'charcoal hana.
- Nenoaio i? Māhele na naau oʻu me ka hui pu ana o paʻakai, a polyethylene glycol pāʻoihana.
- Intravenous? Eaia "MCP" a me "Ondansetron" me ia symptoms o ka nausea a me ka luaʻi.
- ? Eaia "benzodiazepines", "Phenobarbital" ( 'ole thiopental paʻakai) a me kaʻike ākea Muscle relaxants ma hanana o ke kāʻili' ana.
"Theophylline": counterparts
Aia i kekahi mauʻano ai 'o kēiaʻano. Ma keia hihia, noonoo i ka i kēia lapaʻauʻia:
- "Teobiolong" ( "Theobilongum").
- "Spofillinretard" "(Spophillin retard").
- "Perfillon" ( "PerphyUon").
- "Neoefrodal" ( "Neo-Efrodal").
- "Franol" ( "Franol").
waho pūnaewele
Ke me ka pauka, a me nā gula'ā'ī ( "theophylline") waiho i loko o ka pouli, maloo wahi. Lākou holopapa ola o elima makahiki. Waho pūnaewele ihoiho E e hana i loko o ka Pahu Hau. I ka Ia manawa ka mea, e ole e paʻahau. Lākou holopapa-ola o eha makahiki.
hopena
e heluhelu ana i ka luna ma hope, i kekahi ke noonoo ai i na mea i ka lāʻau 'e like me "theophylline", ke kumukuai o ka i mea oluolu ia (i loko o 70-160 hamo i.). Nō hoʻi i loko o kēia kikokikona hai no na olelo ao no ka hoʻohana ana i ka lāʻau a me kona AaOIeIOUIeXAOAaIN me kekahi 'ano.
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